Meptazinol Hydrochloride (CAS 59263-76-2) Suppliers and Product Information

Meptazinol hydrochloride is a centrally active opioid ***gesic. It is a partial agonist at the μ1 opioid receptor and has been shown to inhibit acetylcholinesterase. It is used for the control of moderate to severe pain. Meptazinol has a low propensity toward respiratory depression and other opiate-like side effects, possibly due to its selective interaction with the mu-1 receptor. It also interacts with central cholinergic receptors, which is somewhat unique for an ***gesic.

Frequently Asked Questions

Q: What are the main uses of Meptazinol hydrochloride?

A: Meptazinol hydrochloride is primarily used as an ***gesic for the control of moderate to severe pain. It is a *** ***gesic with antagonist properties, similar in potency to meperidine.

Q: What are the advantages of Meptazinol over other opiates?

A: Meptazinol has a reduced capacity to cause addiction and respiratory depression compared to other opiates. This is due to its intrinsic activity as a partial agonist at the μ1 opioid receptor.

Q: Does Meptazinol have any other notable properties?

A: Yes, Meptazinol has been found to have additional activity as an acetylcholinesterase (AChE) inhibitor, particularly in its ( )-enantiomeric form. This property may partially explain its ***gesic effects and has generated interest in its potential use for treating Alzheimer's disease.